Read Books Online and Download eBooks, EPub, PDF, Mobi, Kindle, Text Full Free.
Download Design And Synthesis Of Peptidomimetic Scaffolds full books in PDF, epub, and Kindle. Read online Design And Synthesis Of Peptidomimetic Scaffolds ebook anywhere anytime directly on your device. Fast Download speed and no annoying ads. We cannot guarantee that every ebooks is available!
Author : Mitchell Huot
Publisher :
ISBN 13 :
Total Pages : pages
Book Rating : 4.:/5 (13 download)
Download or read book Design and Synthesis of Peptidomimetic Scaffolds written by Mitchell Huot and published by . This book was released on 2010 with total page pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Antonio Guarna
Publisher : John Wiley & Sons
ISBN 13 : 1118683145
Total Pages : 334 pages
Book Rating : 4.1/5 (186 download)
Download or read book Peptidomimetics in Organic and Medicinal Chemistry written by Antonio Guarna and published by John Wiley & Sons. This book was released on 2014-03-14 with total page 334 pages. Available in PDF, EPUB and Kindle. Book excerpt: A peptidomimetic is a small protein-like chain designed to mimic a peptide with adjusted molecular properties such as enhanced stability or biological activity. It is a very powerful approach for the generation of small-molecule-based drugs as enzyme inhibitors or receptor ligands. Peptidomimetics in Organic and Medicinal Chemistry outlines the concepts and synthetic strategies underlying the building of bioactive compounds of a peptidomimetic nature. Topics covered include the chemistry of unnatural amino acids, peptide- and scaffold-based peptidomimetics, amino acid-side chain isosteres, backbone isosteres, dipeptide isosteres, beta-turn peptidomimetics, proline-mimetics as turn inducers, cyclic scaffolds, amino acid surrogates, and scaffolds for combinatorial chemistry of peptidomimetics. Case studies in the hit-to-lead process, such as the development of integrin ligands and thrombin inhibitors, illustrate the successful application of peptidomimetics in drug discovery.
Author : Mitchell Huot
Publisher :
ISBN 13 :
Total Pages : pages
Book Rating : 4.:/5 (692 download)
Download or read book Design and Synthesis of Bicyclic Peptidomimetic Scaffolds written by Mitchell Huot and published by . This book was released on 2010 with total page pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Aaron R. Minter
Publisher :
ISBN 13 :
Total Pages : 410 pages
Book Rating : 4.3/5 (91 download)
Download or read book Towards the Design, Synthesis, and Structural Characteristics of Peptidomimetic Scaffolds written by Aaron R. Minter and published by . This book was released on 2005 with total page 410 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Sergey Nicholaevitch Savinov
Publisher :
ISBN 13 :
Total Pages : 610 pages
Book Rating : 4.:/5 (819 download)
Download or read book Design, Synthesis and Application of a Hetero-bicycle-based Peptidomimetic Scaffold written by Sergey Nicholaevitch Savinov and published by . This book was released on 2000 with total page 610 pages. Available in PDF, EPUB and Kindle. Book excerpt:
![Download The Design and Synthesis of Non-peptide Peptidomimetics Based on the [beta]-D-glucose Scaffold and the Development of Rigid Tricyclic Biological Platforms for Ligand Design PDF Online Free](https://books.google.com/books/content/images/frontcover/_5dLNwAACAAJ?fife=w200-h370)
Author : John Hynes
Publisher :
ISBN 13 :
Total Pages : 603 pages
Book Rating : 4.:/5 (187 download)
Download or read book The Design and Synthesis of Non-peptide Peptidomimetics Based on the [beta]-D-glucose Scaffold and the Development of Rigid Tricyclic Biological Platforms for Ligand Design written by John Hynes and published by . This book was released on 1996 with total page 603 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Leonardo Ciofi
Publisher :
ISBN 13 :
Total Pages : pages
Book Rating : 4.:/5 (955 download)
Download or read book Diversity-oriented Synthesis of Peptidomimetic and Natural-product Like Scaffolds written by Leonardo Ciofi and published by . This book was released on 2013* with total page pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Stina Saitton
Publisher :
ISBN 13 : 9789162865245
Total Pages : 70 pages
Book Rating : 4.8/5 (652 download)
Download or read book Design and Synthesis of a Tripeptidomimetic Scaffold Based on Pyridine written by Stina Saitton and published by . This book was released on 2005 with total page 70 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Shawn Earle Richard Schiller
Publisher :
ISBN 13 :
Total Pages : 304 pages
Book Rating : 4.:/5 (433 download)
Download or read book Design and Synthesis of Nuclear Localization Sequence Peptidomimetics Utilizing Glycoside Scaffolding written by Shawn Earle Richard Schiller and published by . This book was released on 1999 with total page 304 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Jaimie K. Rueter
Publisher :
ISBN 13 :
Total Pages : 502 pages
Book Rating : 4.:/5 (318 download)
Download or read book The Design and Synthesis of Peptidomimetics for the Study of Biological Activity written by Jaimie K. Rueter and published by . This book was released on 1998 with total page 502 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Andrea Bordessa
Publisher :
ISBN 13 :
Total Pages : 500 pages
Book Rating : 4.:/5 (495 download)
Download or read book Design, Synthesis and Structural Evaluation of Peptidomimetics Towards Foldamers, PNAs and Non Covalent Inhibitors of the 20S Proteasome written by Andrea Bordessa and published by . This book was released on 2008 with total page 500 pages. Available in PDF, EPUB and Kindle. Book excerpt: The first part of the project at the university of Regensburg, consisted in a stereoselective synthesis of sugar-like d-amino acid. This amino acid was a suitable building block for the synthesis of a-d-oligopeptides containing a sequence of Phe and our building block. Conformational studies of these peptides showed the ability of our building block to induce a secondary structure in the synthesised a-d-peptides, in particular an extended helix structure. In addition, the same furanoic scaffold, has been used for the synthesis of some PNA precursor containing thymine and adenine as nucleobases. The second part of the project at the university of Paris Sud, consisted in the synthesis of peptidomimetics as non covalent inhibitors of 20S proteasome. With the help of molecular modelling, using docking methodology, a small library of molecules was designed: the most promising molecules were then synthesised, showing an inhibitory activity of the proteasome in a micromolar range.
Author : Natasha Susan Murphy
Publisher :
ISBN 13 :
Total Pages : 0 pages
Book Rating : 4.:/5 (883 download)
Download or read book Design and Synthesis of Novel Proteomimetic Scaffolds for the Inhibition of Protein-protein Interactions written by Natasha Susan Murphy and published by . This book was released on 2013 with total page 0 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Thuy-Anh Tran
Publisher :
ISBN 13 :
Total Pages : 576 pages
Book Rating : 4.:/5 (318 download)
Download or read book The Design and Synthesis of Peptidomimetics of Pharmacological Interest written by Thuy-Anh Tran and published by . This book was released on 1997 with total page 576 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Eric Marsault
Publisher : John Wiley & Sons
ISBN 13 : 1119092566
Total Pages : 617 pages
Book Rating : 4.1/5 (19 download)
Download or read book Practical Medicinal Chemistry with Macrocycles written by Eric Marsault and published by John Wiley & Sons. This book was released on 2017-09-12 with total page 617 pages. Available in PDF, EPUB and Kindle. Book excerpt: Including case studies of macrocyclic marketed drugs and macrocycles in drug development, this book helps medicinal chemists deal with the synthetic and conceptual challenges of macrocycles in drug discovery efforts. Provides needed background to build a program in macrocycle drug discovery –design criteria, macrocycle profiles, applications, and limitations Features chapters contributed from leading international figures involved in macrocyclic drug discovery efforts Covers design criteria, typical profile of current macrocycles, applications, and limitations
Author : Matej Živec
Publisher :
ISBN 13 :
Total Pages : 154 pages
Book Rating : 4.:/5 (78 download)
Download or read book Design and synthesis of peptidomimetic inhibitors of peptydoglycan biosynthesis written by Matej Živec and published by . This book was released on 2010 with total page 154 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Joanna Duncan
Publisher :
ISBN 13 :
Total Pages : 544 pages
Book Rating : 4.:/5 (11 download)
Download or read book Design and Synthesis and Testing of Conformationally Constrained Peptidomimetics written by Joanna Duncan and published by . This book was released on 2013 with total page 544 pages. Available in PDF, EPUB and Kindle. Book excerpt:
Author : Claudia Mannino
Publisher :
ISBN 13 :
Total Pages : pages
Book Rating : 4.:/5 (14 download)
Download or read book Design and Synthesis of New Molecular Scaffolds and Their Application as Enzyme Inhibitors written by Claudia Mannino and published by . This book was released on 2008 with total page pages. Available in PDF, EPUB and Kindle. Book excerpt:
